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Human PFKFB3 in complex with a N-Aryl 6-Aminoquinoxaline inhibitor 1

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Protein Data Bank Japan2024-05-15 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6hvh
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Human PFKFB3 in complex with a N-Aryl 6-Aminoquinoxaline inhibitor 1 Descriptor: 3-[[8-(1-methylindol-6-yl)quinoxalin-6-yl]amino]-~{N}-(oxan-4-yl)pyridine-4-carboxamide, 6-O-phosphono-beta-D-fructofuranose, 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3, ... Authors: Banaszak, K, Jakubiec, K, Bialas, A, Fabritius, C.H, Nowak, M. Deposit date: 2018-10-11 Release date: 2018-11-14 Last modified: 2024-05-15 Method: X-RAY DIFFRACTION (2.36 Å) Cite: Discovery and Structure-Activity Relationships of N-Aryl 6-Aminoquinoxalines as Potent PFKFB3 Kinase Inhibitors. ChemMedChem, 14, 2019
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2018-10-11
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