M. thermoresistible GuaB2 delta-CBS in complex with inhibitor Compound 14 (VCC900455)
收藏Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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M. thermoresistible GuaB2 delta-CBS in complex with inhibitor Compound 14 (VCC900455) Descriptor: INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase,Inosine-5'-monophosphate dehydrogenase, cycloheptyl{4-[(isoquinolin-5-yl)sulfonyl]piperazin-1-yl}methanone Authors: Ascher, D.B, Pacitto, A, Blundell, T.L. Deposit date: 2018-04-18 Release date: 2019-05-01 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (1.71 Å) Cite: Synthesis and Structure-Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH. Eur.J.Med.Chem., 174, 2019
创建时间:
2018-04-18



