Co-complex CYP46A1 with 7742 (Soticlestat/TAK-935))
收藏Protein Data Bank Japan2023-10-18 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7lrl
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Co-complex CYP46A1 with 7742 (Soticlestat/TAK-935)) Descriptor: Cholesterol 24-hydroxylase, PROTOPORPHYRIN IX CONTAINING FE, [4-oxidanyl-4-(phenylmethyl)piperidin-1-yl]-(2-pyridin-4-ylpyridin-3-yl)methanone Authors: Lane, W, Yano, J. Deposit date: 2021-02-16 Release date: 2021-08-25 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.995 Å) Cite: Discovery of Soticlestat, a Potent and Selective Inhibitor for Cholesterol 24-Hydroxylase (CH24H). J.Med.Chem., 64, 2021
创建时间:
2021-02-16



