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The STK17A (DRAK1) Kinase Domain Bound to CK156

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Protein Data Bank Japan2024-01-31 更新2026-04-19 收录
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The STK17A (DRAK1) Kinase Domain Bound to CK156 Descriptor: Serine/threonine-protein kinase 17A, ~{N}-~{tert}-butyl-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide Authors: Mathea, S, Preuss, F, Chatterjee, D, Dederer, V, Kurz, C, Hanke, T, Knapp, S. Deposit date: 2022-01-17 Release date: 2022-02-02 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Illuminating the Dark: Highly Selective Inhibition of Serine/Threonine Kinase 17A with Pyrazolo[1,5- a ]pyrimidine-Based Macrocycles. J.Med.Chem., 65, 2022
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2022-01-17
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