five

TEAD2 bound to GNE-7883

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Protein Data Bank Japan2023-10-25 更新2026-04-19 收录
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TEAD2 bound to GNE-7883 Descriptor: (8S)-5-(4-cyclohexylphenyl)-3-[3-(fluoromethyl)azetidine-1-carbonyl]-2-(3-methylpyrazin-2-yl)pyrazolo[1,5-a]pyrimidin-7(4H)-one, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Transcriptional enhancer factor TEF-4 Authors: Noland, C.L, Fong, R. Deposit date: 2022-02-14 Release date: 2023-05-03 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.6 Å) Cite: Novel mechanism of YAP-TEAD inhibition results in targeted chromatin remodeling and reveals an expanded Hippo dependent landscape in cancers To Be Published
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2022-02-14
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