CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c13c(cc(s1)C(NCC2OCCC2)=O)c(nn3c4ccc(cc4)Cl)C, micromolar IC50=0.217
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CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c13c(cc(s1)C(NCC2OCCC2)=O)c(nn3c4ccc(cc4)Cl)C, micromolar IC50=0.217 Descriptor: 1-(4-chlorophenyl)-3-methyl-~{N}-[[(2~{R})-oxolan-2-yl]methyl]thieno[2,3-c]pyrazole-5-carboxamide, GLYCEROL, MAGNESIUM ION, ... Authors: Joseph, C, Rudolph, M.G. Deposit date: 2015-10-21 Release date: 2016-03-09 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.2 Å) Cite: A Real-World Perspective on Molecular Design. J.Med.Chem., 59, 2016
创建时间:
2015-10-21



