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Crystal Structure of human Ser/Thr kinase Pim1 in complex with mitoxantrone

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Protein Data Bank Japan2024-11-27 更新2026-03-21 收录
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Crystal Structure of human Ser/Thr kinase Pim1 in complex with mitoxantrone Descriptor: 1,4-DIHYDROXY-5,8-BIS({2-[(2-HYDROXYETHYL)AMINO]ETHYL}AMINO)-9,10-ANTHRACENEDIONE, Serine/threonine-protein kinase pim-1 Authors: Zhang, W, Wan, X, Xie, Y, Huang, N. Deposit date: 2012-11-27 Release date: 2013-12-11 Last modified: 2024-11-27 Method: X-RAY DIFFRACTION (2.7 Å) Cite: A new target for an old drug: identifying mitoxantrone as a nanomolar inhibitor of PIM1 kinase via kinome-wide selectivity modeling. J. Med. Chem., 56, 2013
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2012-11-27
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