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Focal Adhesion Kinase catalytic domain in complex with irreversible inhibitor

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6gcw
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Focal Adhesion Kinase catalytic domain in complex with irreversible inhibitor Descriptor: 2-[[5-chloranyl-2-[[4-[[[1-[2-(propanoylamino)ethyl]-1,2,3-triazol-4-yl]methylamino]methyl]phenyl]amino]pyrimidin-4-yl]amino]-~{N}-methyl-benzamide, Focal adhesion kinase 1, SULFATE ION Authors: Yen-Pon, E, Li, B, Acebron-Garcia-de-Eulate, M, Tomkiewicz-Raulet, C, Dawson, J, Lietha, D, Frame, M.C, Coumoul, X, Garbay, C, Etheve-Quelquejeu, M, Chen, H. Deposit date: 2018-04-19 Release date: 2019-05-01 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2 Å) Cite: Structure-Based Design, Synthesis, and Characterization of the First Irreversible Inhibitor of Focal Adhesion Kinase. Acs Chem.Biol., 13, 2018
创建时间:
2018-04-19
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