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Cryo-EM structure of CAK in complex with inhibitor BS-194

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Protein Data Bank Japan2024-11-06 更新2026-05-23 收录
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https://pdbj.org/mine/summary/8p6x
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Cryo-EM structure of CAK in complex with inhibitor BS-194 Descriptor: (2S,3S)-3-{[7-(benzylamino)-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-5-yl]amino}butane-1,2,4-triol, CDK-activating kinase assembly factor MAT1, Cyclin-H, ... Authors: Cushing, V.I, Koh, A.F, Feng, J, Jurgaityte, K, Bahl, A.K, Ali, S, Kotecha, A, Greber, B.J. Deposit date: 2023-05-30 Release date: 2024-03-20 Last modified: 2024-11-06 Method: ELECTRON MICROSCOPY (1.9 Å) Cite: High-resolution cryo-EM of the human CDK-activating kinase for structure-based drug design. Nat Commun, 15, 2024
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2023-05-30
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