five

BRD2 Bromodomain2 with A-1360579

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Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5uew
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BRD2 Bromodomain2 with A-1360579 Descriptor: Bromodomain-containing protein 2, N-[3-(4-methoxy-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-4-phenoxyphenyl]methanesulfonamide Authors: Park, C.H. Deposit date: 2017-01-03 Release date: 2017-05-10 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (1.83 Å) Cite: Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors. J. Med. Chem., 60, 2017
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2017-01-03
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