five

The FK1 domain of FKBP51 in complex with SAFit-analog 23c

收藏
Protein Data Bank Japan2024-09-11 更新2026-05-23 收录
下载链接:
https://pdbj.org/mine/summary/9eud
下载链接
链接失效反馈
官方服务:
资源简介:
The FK1 domain of FKBP51 in complex with SAFit-analog 23c Descriptor: (1-propan-2-ylpyrazol-4-yl)methyl (2S)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)ethanoyl]piperidine-2-carboxylate, Peptidyl-prolyl cis-trans isomerase FKBP5 Authors: Meyners, C, Buffa, V, Hausch, F. Deposit date: 2024-03-27 Release date: 2024-06-12 Last modified: 2024-09-11 Method: X-RAY DIFFRACTION (2.022 Å) Cite: 1,4-Pyrazolyl-Containing SAFit-Analogues are Selective FKBP51 Inhibitors With Improved Ligand Efficiency and Drug-Like Profile. Chemmedchem, 19, 2024
创建时间:
2024-03-27
5,000+
优质数据集
54 个
任务类型
进入经典数据集
二维码
社区交流群

面向社区/商业的数据集话题

二维码
科研交流群

面向高校/科研机构的开源数据集话题

数据驱动未来

携手共赢发展

商业合作