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Human Polycomb Repressive Complex 2 in complex with GSK126 inhibitor

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Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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Human Polycomb Repressive Complex 2 in complex with GSK126 inhibitor Descriptor: 1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]-3-methyl-6-[6-(piperazin-1-yl)pyridin-3-yl]-1H-indole-4-carboxamide, Histone-lysine N-methyltransferase EZH2,Polycomb protein SUZ12 (E.C.2.1.1.43) chimera, Polycomb protein EED, ... Authors: Bratkowski, M.A, Liu, X. Deposit date: 2017-07-13 Release date: 2018-06-27 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (3.901 Å) Cite: An Evolutionarily Conserved Structural Platform for PRC2 Inhibition by a Class of Ezh2 Inhibitors. Sci Rep, 8, 2018

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2017-07-13
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