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Crystal structure of the human BRPF1 bromodomain in complex with BZ097

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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Crystal structure of the human BRPF1 bromodomain in complex with BZ097 Descriptor: NITRATE ION, Peregrin, ~{N}-[1,4-dimethyl-2,3-bis(oxidanylidene)-7-pyrrolidin-1-yl-quinoxalin-6-yl]-4-(2-methylpropyl)benzenesulfonamide Authors: Zhu, J, Caflisch, A. Deposit date: 2017-08-28 Release date: 2018-06-27 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Structure-based discovery of selective BRPF1 bromodomain inhibitors. Eur J Med Chem, 155, 2018

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2017-08-28
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