Bromodomain of CBP liganded with BMS-536924 and SGC-CBP30
收藏Protein Data Bank Japan2023-10-25 更新2026-04-19 收录
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Bromodomain of CBP liganded with BMS-536924 and SGC-CBP30 Descriptor: (3M)-4-{[(2S)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-3-[4-methyl-6-(morpholin-4-yl)-1H-benzimidazol-2-yl]pyridin-2(1H)-one, 2-[2-(3-chloro-4-methoxyphenyl)ethyl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[(2S)-2-(morpholin-4-yl)propyl]-1H-benzimidazole, Histone acetyltransferase Authors: Schonbrunn, E, Bikowitz, M. Deposit date: 2022-03-24 Release date: 2023-04-12 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.5 Å) Cite: Structural basis of CBP and EP300 interaction with kinase inhibitors To Be Published
创建时间:
2022-03-24



