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Crystal structure of human ROR gamma LBD in complex with a (quinolinoxymethyl)benzamide inverse agonist

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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Crystal structure of human ROR gamma LBD in complex with a (quinolinoxymethyl)benzamide inverse agonist Descriptor: (2~{S})-1-[2,4-bis(chloranyl)-3-[[2-methyl-4-(trifluoromethyl)quinolin-8-yl]oxymethyl]phenyl]carbonyl-~{N}-methyl-pyrrolidine-2-carboxamide, Nuclear receptor ROR-gamma Authors: Amaudrut, J, Argiriadi, M.A, Barth, M, Breinlinger, E.C, Calderwood, D.J, Cusack, K.P, Kort, M.E, Montalbetti, C, Potin, D, Poupardin, O, Spitzer, L. Deposit date: 2019-08-21 Release date: 2020-09-09 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.2 Å) Cite: Crystal structure of human ROR gamma LBD in complex with a (quinolinoxymethyl)benzamide inverse agonist To Be Published

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2019-08-21
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