Structure of Pi3K gamma with a potent inhibitor: GSK2126458
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Structure of Pi3K gamma with a potent inhibitor: GSK2126458 Descriptor: 2,4-difluoro-N-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamide, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, SULFATE ION Authors: Elkins, P.A, Marrero, E.M. Deposit date: 2009-12-09 Release date: 2010-06-23 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Discovery of GSK2126458, a Highly Potent Inhibitor of PI3K and the Mammalian Target of Rapamycin. ACS Med Chem Lett, 1, 2010
创建时间:
2009-12-09



