PDK1 mutant bound to allosteric disulfide fragment inhibitor 1F8
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https://pdbj.org/mine/summary/3orx
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PDK1 mutant bound to allosteric disulfide fragment inhibitor 1F8 Descriptor: 2-methyl-N-(2-sulfanylethyl)-1-benzofuran-3-carboxamide, 3-phosphoinositide-dependent protein kinase 1, CHLORIDE ION Authors: Sadowsky, J.D, Wells, J.A. Deposit date: 2010-09-08 Release date: 2011-03-23 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.2044 Å) Cite: Turning a protein kinase on or off from a single allosteric site via disulfide trapping. Proc.Natl.Acad.Sci.USA, 108, 2011
创建时间:
2010-09-08



