five

Bromodomain of CBP liganded with inhibitor iCBP5

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Protein Data Bank Japan2024-05-08 更新2026-04-19 收录
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https://pdbj.org/mine/summary/8ga2
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资源简介:
Bromodomain of CBP liganded with inhibitor iCBP5 Descriptor: (6S)-6-{(5M)-5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[(1s,4R)-4-methoxycyclohexyl]-1H-benzimidazol-2-yl}-1-phenylpiperidin-2-one, 1,2-ETHANEDIOL, CREB-binding protein Authors: Schonbrunn, E, Bikowitz, M. Deposit date: 2023-02-22 Release date: 2024-02-28 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Group 3 medulloblastoma transcriptional networks collapse under domain specific EP300/CBP inhibition. Nat Commun, 15, 2024
创建时间:
2023-02-22
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