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Peptide-Based Inhibitors of Plk1 Polo-box Domain

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Protein Data Bank Japan2025-03-26 更新2026-03-21 收录
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Peptide-Based Inhibitors of Plk1 Polo-box Domain Descriptor: Peptide-Based inhibitor, Serine/threonine-protein kinase PLK1 Authors: Qian, W.-J, Park, J.-E, Lim, D.C, Park, S.-Y, Lee, K.-W, Yaffe, M.B, Lee, K.S, Burke, T.R. Deposit date: 2013-12-23 Release date: 2014-12-03 Last modified: 2025-03-26 Method: X-RAY DIFFRACTION (1.448 Å) Cite: Mono-anionic phosphopeptides produced by unexpected histidine alkylation exhibit high plk1 polo-box domain-binding affinities and enhanced antiproliferative effects in hela cells. Biopolymers, 102, 2014

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2013-12-23
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