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Aurora-A Inhibitor Structure (2nd crystal form)

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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Aurora-A Inhibitor Structure (2nd crystal form) Descriptor: 4-{[9-CHLORO-7-(2,6-DIFLUOROPHENYL)-5H-PYRIMIDO[5,4-D][2]BENZAZEPIN-2-YL]AMINO}BENZOIC ACID, SERINE/THREONINE-PROTEIN KINASE 6 AURORA/IPL1-RELATED KINASE 1, BREAST TUMOR-AMPLIFIED KINASE, ... Authors: Kosmopoulou, M, Bayliss, R. Deposit date: 2009-09-24 Release date: 2010-01-26 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (3.302 Å) Cite: Crystal Structure of an Aurora-A Mutant that Mimics Aurora-B Bound to Mln8054: Insights Into Selectivity and Drug Design. Biochem.J., 427, 2010
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2009-09-24
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