遇见数据集

Leishmania major N-myristoyltransferase in complex with quinazoline inhibitor IMP-0000811

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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Leishmania major N-myristoyltransferase in complex with quinazoline inhibitor IMP-0000811 Descriptor: 3-[methyl-[2-[methyl-(1-methylpiperidin-4-yl)amino]quinazolin-4-yl]amino]propanenitrile, Glycylpeptide N-tetradecanoyltransferase, MAGNESIUM ION, ... Authors: Brannigan, J.A. Deposit date: 2019-01-01 Release date: 2020-05-06 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.6 Å) Cite: Novel Thienopyrimidine Inhibitors of Leishmania N -Myristoyltransferase with On-Target Activity in Intracellular Amastigotes. J.Med.Chem., 63, 2020

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2019-01-01
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