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Aurora kinase selective inhibitors identified using a Taxol-induced checkpoint sensitivity screen.

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Aurora kinase selective inhibitors identified using a Taxol-induced checkpoint sensitivity screen. Descriptor: 2-((4-(4-HYDROXYPIPERIDIN-1-YL)PHENYL)AMINO)-5,11-DIMETHYL-5H-BENZO[E]PYRIMIDO [5,4-B][1,4]DIAZEPIN-6(11H)-ONE, INNER CENTROMERE PROTEIN A, SERINE/THREONINE-PROTEIN KINASE 12-A Authors: Kwiatkowski, N, Villa, F, Musacchio, A, Gray, N. Deposit date: 2011-07-12 Release date: 2012-02-01 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Selective Aurora Kinase Inhibitors Identified Using a Taxol- Induced Checkpoint Sensitivity Screen. Acs Chem.Biol., 7, 2012

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2011-07-12
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