Mutated Mus Musculus P38 Kinase (mP38)
收藏Protein Data Bank Japan2023-08-23 更新2026-03-21 收录
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https://pdbj.org/mine/summary/1yw2
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Mutated Mus Musculus P38 Kinase (mP38) Descriptor: 2-(ETHOXYMETHYL)-4-(4-FLUOROPHENYL)-3-[2-(2-HYDROXYPHENOXY)PYRIMIDIN-4-YL]ISOXAZOL-5(2H)-ONE, Mitogen-activated protein kinase 14 Authors: Laughlin, S.K, Clark, M.P, Djung, J.F, Golebiowski, A, Brugel, T.A, Sabat, M, Bookland, R.G, Laufersweiler, M.J, Vanrens, J.C, Townes, J.A, De, B, Hsieh, L.C, Xu, S.C, Walter, R.L, Mekel, M.J, Janusz, M.J. Deposit date: 2005-02-16 Release date: 2005-05-10 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (2.01 Å) Cite: The development of new isoxazolone based inhibitors of tumor necrosis factor-alpha (TNF-alpha) production. Bioorg.Med.Chem.Lett., 15, 2005
创建时间:
2005-02-16



