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Crystal structure of human liver FBPase complexed with an covalent inhibitor

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Protein Data Bank Japan2024-10-23 更新2026-04-19 收录
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Crystal structure of human liver FBPase complexed with an covalent inhibitor Descriptor: 1,2-BENZISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDE, ADENOSINE MONOPHOSPHATE, Fructose-1,6-bisphosphatase 1, ... Authors: Cao, H, Huang, Y, Ren, Y, Wan, J. Deposit date: 2022-01-08 Release date: 2022-07-13 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (1.724 Å) Cite: N -Acylamino Saccharin as an Emerging Cysteine-Directed Covalent Warhead and Its Application in the Identification of Novel FBPase Inhibitors toward Glucose Reduction. J.Med.Chem., 65, 2022

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2022-01-08
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