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Structure of NEDD8-activating enzyme in complex with NEDD8 and MLN4924

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Structure of NEDD8-activating enzyme in complex with NEDD8 and MLN4924 Descriptor: NEDD8, NEDD8-activating enzyme E1 catalytic subunit, NEDD8-activating enzyme E1 regulatory subunit, ... Authors: Sintchak, M.D. Deposit date: 2009-04-07 Release date: 2010-02-02 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (3 Å) Cite: Substrate-assisted inhibition of ubiquitin-like protein-activating enzymes: the NEDD8 E1 inhibitor MLN4924 forms a NEDD8-AMP mimetic in situ. Mol.Cell, 37, 2010

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2009-04-07
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