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Crystal structure of K103N/Y181C mutant HIV-1 reverse transcriptase (RT) in complex with TMC278 (Rilpivirine), a non-nucleoside RT inhibitor

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Protein Data Bank Japan2023-11-01 更新2026-03-21 收录
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Crystal structure of K103N/Y181C mutant HIV-1 reverse transcriptase (RT) in complex with TMC278 (Rilpivirine), a non-nucleoside RT inhibitor Descriptor: 1,2-ETHANEDIOL, 4-{[4-({4-[(E)-2-cyanoethenyl]-2,6-dimethylphenyl}amino)pyrimidin-2-yl]amino}benzonitrile, Reverse transcriptase/ribonuclease H, ... Authors: Das, K, Bauman, J.D, Clark Jr, A.D, Shatkin, A.J, Arnold, E. Deposit date: 2007-11-27 Release date: 2008-02-12 Last modified: 2023-11-01 Method: X-RAY DIFFRACTION (2.1 Å) Cite: High-resolution structures of HIV-1 reverse transcriptase/TMC278 complexes: Strategic flexibility explains potency against resistance mutations. Proc.Natl.Acad.Sci.Usa, 105, 2008
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2007-11-27
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