five

Co-crystal structure of BTK kinase domain with inhibitor

收藏
Protein Data Bank Japan2024-11-13 更新2026-04-25 收录
下载链接:
https://pdbj.org/mine/summary/7yc9
下载链接
链接失效反馈
官方服务:
资源简介:
Co-crystal structure of BTK kinase domain with inhibitor Descriptor: (7~{S})-2-(4-bromanyl-3,5-dimethoxy-phenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide, 1,2-ETHANEDIOL, Tyrosine-protein kinase BTK Authors: Zhou, X. Deposit date: 2022-07-01 Release date: 2023-05-17 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.4 Å) Cite: Discovery of BGB-8035, a Highly Selective Covalent Inhibitor of Bruton's Tyrosine Kinase for B-Cell Malignancies and Autoimmune Diseases. J.Med.Chem., 66, 2023
创建时间:
2022-07-01
5,000+
优质数据集
54 个
任务类型
进入经典数据集
二维码
社区交流群

面向社区/商业的数据集话题

二维码
科研交流群

面向高校/科研机构的开源数据集话题

数据驱动未来

携手共赢发展

商业合作