遇见数据集

PXR IN COMPLEX WITH THROMBIN INHIBITOR COMPOUND 17

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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PXR IN COMPLEX WITH THROMBIN INHIBITOR COMPOUND 17 Descriptor: (4S)-2-METHYL-2,4-PENTANEDIOL, DIMETHYL SULFOXIDE, GLYCEROL, ... Authors: Hillig, R.C, Puetter, V. Deposit date: 2019-11-14 Release date: 2020-11-11 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Design, Synthesis, and Pharmacological Characterization of a Neutral, Non-Prodrug Thrombin Inhibitor with Good Oral Pharmacokinetics. J.Med.Chem., 63, 2020

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2019-11-14
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