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Crystal structure of TNKS2 in complex with 2-(4-chlorophenyl)-1,2,3,4- tetrahydroquinazolin-4-one

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Crystal structure of TNKS2 in complex with 2-(4-chlorophenyl)-1,2,3,4- tetrahydroquinazolin-4-one Descriptor: (2S)-2-(4-chlorophenyl)-2,3-dihydro-1H-quinazolin-4-one, GLYCEROL, SULFATE ION, ... Authors: Nkizinkiko, Y, Lehtio, L. Deposit date: 2015-03-05 Release date: 2015-07-29 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.07 Å) Cite: Discovery of Potent and Selective Nonplanar Tankyrase Inhibiting Nicotinamide Mimics. Bioorg.Med.Chem., 23, 2015
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2015-03-05
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