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Crystal Structure Of AKR1B10 Complexed With NADP+ And Epalrestat

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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Crystal Structure Of AKR1B10 Complexed With NADP+ And Epalrestat Descriptor: Aldo-keto reductase family 1 member B10, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, {5-[(2E)-2-methyl-3-phenylprop-2-en-1-ylidene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl}acetic acid Authors: Zhang, L, Zheng, X, Zhang, H, Zhao, Y, Chen, K, Zhai, J, Hu, X, Structural Genomics Consortium (SGC) Deposit date: 2013-03-06 Release date: 2013-10-23 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Inhibitor selectivity between aldo-keto reductase superfamily members AKR1B10 and AKR1B1: Role of Trp112 (Trp111). Febs Lett., 587, 2013
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2013-03-06
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