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Crystal structure of aminoglycoside resistance enzyme ApmA, complex with gentamicin

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Protein Data Bank Japan2026-02-25 更新2026-04-19 收录
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Crystal structure of aminoglycoside resistance enzyme ApmA, complex with gentamicin Descriptor: (2R,3R,4R,5R)-2-((1S,2S,3R,4S,6R)-4,6-DIAMINO-3-((2R,3R,6S)-3-AMINO-6-(AMINOMETHYL)-TETRAHYDRO-2H-PYRAN-2-YLOXY)-2-HYDR OXYCYCLOHEXYLOXY)-5-METHYL-4-(METHYLAMINO)-TETRAHYDRO-2H-PYRAN-3,5-DIOL, 1,2-ETHANEDIOL, Aminocyclitol acetyltransferase ApmA, ... Authors: Stogios, P.J, Evdokimova, E, Osipiuk, J, Di Leo, R, Bordeleau, E, Wright, G.D, Savchenko, A, Joachimiak, A, Satchell, K.J.F, Center for Structural Biology of Infectious Diseases (CSBID) Deposit date: 2022-04-28 Release date: 2023-04-19 Last modified: 2026-02-25 Method: X-RAY DIFFRACTION (1.78 Å) Cite: Mechanistic plasticity in ApmA enables aminoglycoside promiscuity for resistance Nat.Chem.Biol., 20, 2024
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2022-04-28
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