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Crystal structure of benzamide 9 bound to AuroraA

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Protein Data Bank Japan2024-02-21 更新2026-03-21 收录
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Crystal structure of benzamide 9 bound to AuroraA Descriptor: N-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamide, cDNA FLJ58295, highly similar to Serine/threonine-protein kinase 6 Authors: Huang, X. Deposit date: 2010-07-27 Release date: 2010-08-18 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (2 Å) Cite: Discovery of a potent, selective, and orally bioavailable pyridinyl-pyrimidine phthalazine aurora kinase inhibitor. J.Med.Chem., 53, 2010

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2010-07-27
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