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Crystal structure of Eis from Mycobacterium tuberculosis in complex with inhibitor SGT1358

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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Crystal structure of Eis from Mycobacterium tuberculosis in complex with inhibitor SGT1358 Descriptor: 2-[(4-amino-6,7,8,9-tetrahydro-5H-cyclohepta[4,5]thieno[2,3-d]pyrimidin-2-yl)sulfanyl]-N-[2-(piperidin-1-yl)ethyl]acetamide, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ... Authors: Punetha, A, Hou, C, Ngo, H.X, Garneau-Tsodikova, S, Tsodikov, O.V. Deposit date: 2020-02-16 Release date: 2020-06-03 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Structure-Guided Optimization of Inhibitors of Acetyltransferase Eis fromMycobacterium tuberculosis. Acs Chem.Biol., 15, 2020
创建时间:
2020-02-16
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