遇见数据集

IRE1 complexed with Cdk1/2 Inhibitor III

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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IRE1 complexed with Cdk1/2 Inhibitor III Descriptor: 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE, Serine/threonine-protein kinase/endoribonuclease IRE1 Authors: Lee, K.P.K, Sicheri, F. Deposit date: 2010-01-25 Release date: 2010-05-12 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (3.33 Å) Cite: Flavonol activation defines an unanticipated ligand-binding site in the kinase-RNase domain of IRE1. Mol.Cell, 38, 2010

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2010-01-25
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