five

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 (3R,4R)-N-cyclohexyl-4-((3-methyl-2-oxo-1,2-dihydro-1,7-naphthyridin-8-yl)amino)piperidine-3-carboxamide

收藏
Protein Data Bank Japan2024-05-01 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/6z7m
下载链接
链接失效反馈
官方服务:
资源简介:
N-TERMINAL BROMODOMAIN OF HUMAN BRD4 (3R,4R)-N-cyclohexyl-4-((3-methyl-2-oxo-1,2-dihydro-1,7-naphthyridin-8-yl)amino)piperidine-3-carboxamide Descriptor: (3R,4R)-N-cyclohexyl-4-((3-methyl-2-oxo-1,2-dihydro-1,7-naphthyridin-8-yl)amino)piperidine-3-carboxamide, Bromodomain-containing protein 4 Authors: Chung, C. Deposit date: 2020-05-31 Release date: 2020-07-29 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.26 Å) Cite: GSK789: A Selective Inhibitor of the First Bromodomains (BD1) of the Bromo and Extra Terminal Domain (BET) Proteins. J.Med.Chem., 63, 2020
创建时间:
2020-05-31
二维码
社区交流群
二维码
科研交流群
商业服务