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Crystal Structure of SARS-CoV-2 Main Protease (Mpro) E166R Mutant in Complex with Inhibitor GC376

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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Crystal Structure of SARS-CoV-2 Main Protease (Mpro) E166R Mutant in Complex with Inhibitor GC376 Descriptor: (1S,2S)-2-({N-[(benzyloxy)carbonyl]-L-leucyl}amino)-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonic acid, 3C-like proteinase nsp5 Authors: Lewandowski, E.M, Chen, Y. Deposit date: 2022-06-18 Release date: 2022-08-31 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.78 Å) Cite: A yeast-based system to study SARS-CoV-2 Mpro structure and to identify nirmatrelvir resistant mutations. Plos Pathog., 19, 2023
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2022-06-18
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