Crystal structure of bromodomain from Plasmodium falciparum GCN5 complexed with a ligand
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Crystal structure of bromodomain from Plasmodium falciparum GCN5 complexed with a ligand Descriptor: CHLORIDE ION, N-[(2S)-3-[2,4-bis(oxidanylidene)pyrimidin-1-yl]-1-(methylamino)-1-oxidanylidene-propan-2-yl]-6-methoxy-3H-imidazo[4,5-b]pyridine-7-carboxamide, histone acetyltransferase Authors: McMillan, J, Postis, V, Masson, G. Deposit date: 2025-12-11 Release date: 2026-04-08 Last modified: 2026-06-10 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Residue-Level Determination of Small-Molecule-Protein Affinities by Hydrogen-Deuterium Exchange Mass Spectrometry. J.Am.Soc.Mass.Spectrom., 37, 2026
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2025-12-11



