Aspartyl/Asparaginyl beta-hydroxylase (AspH) oxygenase and TPR domains in complex with manganese, 3-fluoropyridine-2,4-dicarboxylic acid, and factor X substrate peptide fragment (39mer-4Ser)
收藏Protein Data Bank Japan2024-11-20 更新2026-04-19 收录
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Aspartyl/Asparaginyl beta-hydroxylase (AspH) oxygenase and TPR domains in complex with manganese, 3-fluoropyridine-2,4-dicarboxylic acid, and factor X substrate peptide fragment (39mer-4Ser) Descriptor: 3-fluoranylpyridine-2,4-dicarboxylic acid, Aspartyl/asparaginyl beta-hydroxylase, Coagulation factor X, ... Authors: Nakashima, Y, Brewitz, L, Schofield, C.J. Deposit date: 2021-01-20 Release date: 2021-06-02 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.66 Å) Cite: Fluorinated derivatives of pyridine-2,4-dicarboxylate are potent inhibitors of human 2-oxoglutarate dependent oxygenases J Fluor Chem, 247, 2021
创建时间:
2021-01-20



