five

N-terminal bromodomain of BRD4 in complex with OTX-015

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Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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N-terminal bromodomain of BRD4 in complex with OTX-015 Descriptor: 1,2-ETHANEDIOL, 4-{6-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[(1S)-1-(pyridin-2-yl)ethyl]-1H-pyrrolo[3,2-b]pyridin-3-yl}benzoic acid, Bromodomain-containing protein 4 Authors: Zhang, Y. Deposit date: 2017-07-28 Release date: 2018-08-01 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (1.19 Å) Cite: BRD4 Profiling Identifies Critical Chronic Lymphocytic Leukemia Oncogenic Circuits and Reveals Sensitivity to PLX51107, a Novel Structurally Distinct BET Inhibitor. Cancer Discov, 8, 2018
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2017-07-28
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