DCN1 bound to DI-591
收藏Protein Data Bank Japan2024-04-03 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5ufi
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DCN1 bound to DI-591 Descriptor: DCN1-like protein 1, N-[(1S)-1-cyclohexyl-2-{[3-(morpholin-4-yl)propanoyl]amino}ethyl]-N~2~-propanoyl-3-[6-(propan-2-yl)-1,3-benzothiazol-2-yl]-L-alaninamide Authors: Stuckey, J. Deposit date: 2017-01-04 Release date: 2017-11-01 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.58 Å) Cite: A potent small-molecule inhibitor of the DCN1-UBC12 interaction that selectively blocks cullin 3 neddylation. Nat Commun, 8, 2017
创建时间:
2017-01-04



