遇见数据集

Notum complex with ARUK3003778

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Notum complex with ARUK3003778 Descriptor: 3-(3,4-dichlorophenyl)sulfanyl-1$l^{4},2,7,8-tetrazabicyclo[4.3.0]nona-1(6),2,4,7-tetraen-9-one, DIMETHYL SULFOXIDE, Palmitoleoyl-protein carboxylesterase NOTUM, ... Authors: Jones, E.Y, Fish, P. Deposit date: 2020-12-03 Release date: 2022-01-12 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.33 Å) Cite: Virtual Screening Directly Identifies New Fragment-Sized Inhibitors of Carboxylesterase Notum with Nanomolar Activity. J.Med.Chem., 65, 2022

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2020-12-03
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