PPARg bound to inverse agonist H3B-343
收藏Protein Data Bank Japan2023-10-25 更新2026-04-19 收录
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https://pdbj.org/mine/summary/8dsy
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PPARg bound to inverse agonist H3B-343 Descriptor: Peroxisome proliferator-activated receptor gamma, {5-[(5-{[(4-tert-butylphenyl)methyl]carbamoyl}-2,3-dimethyl-1H-indol-1-yl)methyl]-2-chlorophenoxy}acetic acid Authors: Larsen, N.A. Deposit date: 2022-07-24 Release date: 2022-09-07 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (2.95 Å) Cite: Biochemical and structural basis for the pharmacological inhibition of nuclear hormone receptor PPAR gamma by inverse agonists. J.Biol.Chem., 298, 2022
创建时间:
2022-07-24



