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BRD4 (BD1) in complex with APSC-derived ligands (e.g. SSLH01 a sulfasalazine derivate)

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6g0h
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BRD4 (BD1) in complex with APSC-derived ligands (e.g. SSLH01 a sulfasalazine derivate) Descriptor: 1,2-ETHANEDIOL, 4-azanyl-2-oxidanyl-5-[(~{E})-[4-(pyridin-2-ylsulfamoyl)phenyl]diazenyl]benzoic acid, Bromodomain-containing protein 4, ... Authors: Humbeck, L, Pretzel, J. Deposit date: 2018-03-18 Release date: 2020-01-08 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.907 Å) Cite: Discovery of an Unexpected Similarity in Ligand Binding Between BRD4 and PPARgamma Chemrxiv, 2019
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2018-03-18
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