EGFR kinase (T790M/L858R) with inhibitor compound 8
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https://pdbj.org/mine/summary/4rj8
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EGFR kinase (T790M/L858R) with inhibitor compound 8 Descriptor: 1-cyclopentyl-N-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1H-pyrrolo[3,2-c]pyridin-6-amine, Epidermal growth factor receptor, SULFATE ION Authors: Eigenbrot, C, Yu, C. Deposit date: 2014-10-08 Release date: 2014-11-26 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (2.5 Å) Cite: Discovery of Selective and Noncovalent Diaminopyrimidine-Based Inhibitors of Epidermal Growth Factor Receptor Containing the T790M Resistance Mutation. J.Med.Chem., 57, 2014
创建时间:
2014-10-08



