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Crystal Structure of SARS-CoV-2 Omicron Main Protease (Mpro) in Complex with Nirmatrelvir

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Protein Data Bank Japan2025-04-09 更新2026-04-04 收录
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https://pdbj.org/mine/summary/8hoz
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Crystal Structure of SARS-CoV-2 Omicron Main Protease (Mpro) in Complex with Nirmatrelvir Descriptor: (1R,2S,5S)-N-{(1E,2S)-1-imino-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl}-6,6-dimethyl-3-[3-methyl-N-(trifluoroacetyl)-L-valyl]-3-azabicyclo[3.1.0]hexane-2-carboxamide, 3C-like proteinase nsp5 Authors: Lin, M, Liu, X. Deposit date: 2022-12-11 Release date: 2023-12-13 Last modified: 2025-04-09 Method: X-RAY DIFFRACTION (2.83 Å) Cite: Molecular mechanism of ensitrelvir inhibiting SARS-CoV-2 main protease and its variants. Commun Biol, 6, 2023
创建时间:
2022-12-11
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