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Human EphA3 kinase domain in complex with inhibitor AWL-II-38.3

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Protein Data Bank Japan2023-08-30 更新2026-03-21 收录
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https://pdbj.org/mine/summary/3dzq
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Human EphA3 kinase domain in complex with inhibitor AWL-II-38.3 Descriptor: EPH receptor A3, N-[2-methyl-5-({[3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamide Authors: Walker, J.R, Syeda, F, Gray, N, Mansoor, W, Mackenzie, F, Bountra, C, Weigelt, J, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC) Deposit date: 2008-07-30 Release date: 2008-08-26 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (1.75 Å) Cite: Kinase Domain of Human Ephrin Type-A Receptor 3 (Epha3) in Complex with ALW-II-38-3. To be Published
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2008-07-30
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