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Crystal structure of Ser/Thr kinase Pim1 in complex with 10-DEBC derivatives

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Protein Data Bank Japan2024-10-09 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6l17
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Crystal structure of Ser/Thr kinase Pim1 in complex with 10-DEBC derivatives Descriptor: 7-chloranyl-5-[3-[(3~{S})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazin-8-amine, Serine/threonine-protein kinase pim-1 Authors: Zhang, W, Xie, Y, Cao, R, Huang, N, Zhou, Y. Deposit date: 2019-09-27 Release date: 2020-09-02 Last modified: 2024-10-09 Method: X-RAY DIFFRACTION (1.75 Å) Cite: Structure-Based Optimization of 10-DEBC Derivatives as Potent and Selective Pim-1 Kinase Inhibitors. J.Chem.Inf.Model., 60, 2020
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2019-09-27
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