Comparison of binding affinities (Ki) of MT1 receptors in CHO and Pichia pastoris (P.p.) membranes, and purified in a 0.1% Fos14/0.1% CHAPS mixture.
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https://figshare.com/articles/dataset/_Comparison_of_binding_affinities_Ki_of_MT1_receptors_in_CHO_and_Pichia_pastoris_P_p_membranes_and_purified_in_a_0_1_Fos14_0_1_CHAPS_mixture_/1082107
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Twenty-four compounds from our MT1 ligands collection were tested. 4P-PDOT, Luzindole, S 22153, D600, S 73893-1, S 77834, and S 77840 are antagonist ligands, while the others are agonist ligands. Concentration-response curves were analyzed by non-linear regression. Binding affinities are expressed as mean pKi ± SEM of four independent experiments.
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2015-12-02



