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Structure of GRP94 with a resorcinylic inhibitor.

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Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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Structure of GRP94 with a resorcinylic inhibitor. Descriptor: 1,2-ETHANEDIOL, 5-[2-(1-benzyl-1H-imidazol-2-yl)ethyl]-4,6-dichlorobenzene-1,3-diol, Endoplasmin, ... Authors: Que, N.L.S, Gewirth, D.T. Deposit date: 2018-01-25 Release date: 2018-04-18 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.895 Å) Cite: Structure Based Design of a Grp94-Selective Inhibitor: Exploiting a Key Residue in Grp94 To Optimize Paralog-Selective Binding. J. Med. Chem., 61, 2018

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2018-01-25
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