Crystal structure of human BRD4(1) bromodomain in complex with DR46
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Crystal structure of human BRD4(1) bromodomain in complex with DR46 Descriptor: Bromodomain-containing protein 4, ~{N}-[3-(5-ethanoyl-2-ethoxy-phenyl)-5-(1-methylpyrazol-3-yl)phenyl]furan-2-carboxamide Authors: Zhu, J, Caflisch, A. Deposit date: 2017-08-28 Release date: 2018-10-10 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Chemical Space Expansion of Bromodomain Ligands Guided by in Silico Virtual Couplings (AutoCouple). Acs Cent.Sci., 4, 2018
创建时间:
2017-08-28



